Current Medicinal Chemistry |
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20 amino acids affinity agents allopurinol amastigotes amino acids Amphotericin analogs antileishmanial antimonials assay bead bead-one Bentham Science Publishers binding biological activity brazi/iensis building blocks carbohydrates carboxylic acids catalysis cells Chem chemical steps combinatorial chemistry combinatorial libraries Couple cutaneous leishmaniasis disease donovani dose drug design drug discovery efficacy encoded enzyme formycin functional groups glucantime hexapeptide inhibiting inhibitors interaction involve isomerization Kala-azar large number Lead Discovery leishmanicidal activity libraries of compounds ligand linker matrix medicinal chemistry metabolic metabolite method methodology molecules motif nucleic acid oligonucleotide oxidation parasite pentavalent antimonial peptide libraries permutational library pharmacophores positions potent Primer produced promastigotes protein RARs recently reported resin retinoic acid retinoid retinol screening selected sequence set of 20 shown small molecule sodium stibogluconate solid phase synthesis specific split synthesis scheme strategy structure sublibraries substrate tags target techniques therapeutic tissue toxic TTNPB visceral leishmaniasis vitamin vitro vivo